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Displacement of [3H]nitrendipine from voltage-dependent calcium channel in rat brain cortex by scintillation counting
Assay data:3 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 3 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed Citation
Inhibition of calcium activation was assessed against calcium-induced constriction of potassium-depolarized rat aorta (Negative logarithm of the molar concentration)
Assay data:36 Active, 1 Activity ≤ 1 nM, 36 Activity ≤ 1 µM, 36 Tested
Inhibition constant by its ability to inhibit (act through Ca++ ion channel) contractions induced by K+ depolarization in rat dorsal aorta
Assay data:6 Active, 1 Activity ≤ 1 nM, 7 Activity ≤ 1 µM, 7 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µM
Inhibition of contractions induced by K+ depolarization in rat dorsal aorta
Assay data:15 Active, 2 Activity ≤ 1 nM, 19 Activity ≤ 1 µM, 19 Tested
Compound was tested for ability to relax potassium-contracted rabbit aorta smooth muscle
Assay data:8 Active, 2 Activity ≤ 1 nM, 7 Activity ≤ 1 µM, 8 Tested
Calcium channel-blocking activity by determined by ability to antagonize calcium-induced contractions of isolated rabbit aortic strips
Assay data:60 Active, 2 Activity ≤ 1 nM, 60 Activity ≤ 1 µM, 60 Tested
Compound was tested for its antagonist activity against calcium channel
Assay data:22 Active, 8 Activity ≤ 1 nM, 22 Activity ≤ 1 µM, 23 Tested
Inhibition of [3H]nitrendipine binding to L-type calcium channel dihydropyridine site of porcine cardiac sarcolemma membrane vesicles
Assay data:12 Active, 3 Activity ≤ 1 nM, 8 Activity ≤ 1 µM, 12 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranes
Assay data:9 Active, 1 Activity ≤ 1 nM, 7 Activity ≤ 1 µM, 14 Tested
Calcium channel blocking activity in rabbit
Assay data:11 Active, 1 Activity ≤ 1 nM, 5 Activity ≤ 1 µM, 13 Tested
Inhibition of [3H]nitrendipine binding to calcium channels in Rabbit cardiac muscle.
Assay data:18 Active, 1 Activity ≤ 1 nM, 6 Activity ≤ 1 µM, 21 Tested
Dissociation constant for inhibition of [3H]nitrendipine binding to guinea pig myocardial membranes
Assay data:8 Active, 5 Activity ≤ 1 nM, 8 Activity ≤ 1 µM, 8 Tested
The compound was tested in vitro for its ability to displace [3H]PN-200-110 from Calcium Channel in rat brain membranes.
Assay data:6 Active, 1 Activity ≤ 1 nM, 17 Activity ≤ 1 µM, 18 Tested
[Ca2+] channel binding affinity was evaluated by its ability to displace [3H]-PN-200-110 in rat brain synaptosomes
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